Burkamp

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Primary tabs

1. Personal Information

Name
Frank Burkamp
Organization(s)
MSD - UK, AstraZeneca - Sweden

2. Community Expertise

The Synaptic Leap community
Skills
Chemistry

3. Publications

Publications

PATENTS

1. Burkamp, F.; Castro Pineiro, J. L.; Hollingworth, G. J.: Prodrugs of substituted amino heterobicycles which modulate the function of the vanilloid-1 receptor (VR1); WO 2005080391 A1 (2005).
2. Bayliss, T.; Brown, R. E.; Burkamp, F.; Jones, A. B.; Neduvelil, J. G.: Preparation of pyridyl-piperidine-carboxamide derivatives as modulators of vanilloid-1 receptor (VR-1); WO 2005041390 A1 (2005).
3. Burkamp, F.; Fletcher, S. R.: Indazol-3-ones and analogs and derivatives which modulate the function of the vanilloid-1 receptor (VR1); WO 2005049601 A1 (2005).
4. Blurton, P.; Burkamp, F.; Fletcher, S. R.; Jones, B. A.; Mciver, E. G.: Preparation of substituted 1-phthalazinamines as vanilloid receptor (VR1) antagonists for treating pain and/ or inflammation; WO 2004099177 A1 (2004).
5. Brown, R. E.; Burkamp, F.; Doughty, V. A.; Fletcher, S. R.; Hollingworth, G. J.; Jones, B. A.; Sparey, T. J.: Preparation of amino heterocycles as vanilliod receptor (VR1) modulators, in particular antagonists, for treating pain and/ or inflammation ; WO 2004074290 A1 (2004).
6. Blurton, P.; Burkamp, F.; Fletcher, S. R.; Hollingworth, G. J.; Jones, A. B.; Mciver, E. G.; Moyes, C. R.; Rogers, L.: Preparation of amino heterocycles as vanilloid receptor (VR1) modulators, in particular antagonists, for treating pain and/ or inflammation; WO 2004046133 A1 (2004).
7. Blackaby, W. P.; Blurton, P.; Burkamp, F.; Fletcher, S. R.; Jennings, A. L.; Richard, T.; MacLeod, A. M.; Street, L. J.; Thomas, S.; Van Niel, M. B.; Wilson, K.: Preparation of phenylpyridazine derivatives as ligands for GABA receptors; WO 2004014865 A1 (2004).
8. Burkamp, F.; Street, L. J. Preparation of imidazo[4,5-b]pyridines as ligands for GABA receptors for treating/ preventing neurological disorders; WO 2003086406 (2003).
9. Blurton, P.; Burkamp, F.; Fletcher, S. R.: Preparation of triazolophthalazines, -quinolines and -isoquinolines as ligands for GABAa receptors containing the 5 subtype; WO 200281474 A1 (2002).
10. Burkamp, F.; Cheng, S. K.-F.; Fletcher, S. R.: Preparation of phenylsulphonylpiperazinyl derivatives as 5-HT receptor ligands; WO 200174797 A1 (2001).
11. Blurton, P.; Burkamp, F.; Cheng, S. K.-F.; Fletcher, S. R.; MacLeod, A. M.; Van Niel, M. B.: Preparation of phenylsulphonyl derivatives as 5-HT receptor ligands; WO 200043362 A1 (2000).

PUBLICATIONS

1. Enders, D.; Burkamp, F.: -Heterosubstituted Aldehydes in Organic Synthesis. Enantioselective Approaches to New Analogues of Mevinic Acids; Collect. Czech. Chem. Commun., 2003; 68(5), 975-1006.
2. Burkamp, F.; Fletcher, S. R.: Preparation of 3-Aminoalkyl-benzo[b]thiophenes; J. Het. Chem. 2002, 39, 1177-1188.

3. Fletcher, S. R.; Burkamp, F.; Blurton, P.; Cheng, S. K.-F.; Clarkson, R.; O'Connor, D.; Spinks, D.; Tudge, M.; van Niel, M. B.; Patel, S.; Chapman, K.; Marwood, R.; Shepheard, S.; Bentley, G.; Cook, G. P.; Bristow, L. J.; Castro, J. L.; Hutson, P. H.; MacLeod, A. M.: 4-(Phenylsulfonyl)piperidines: Novel, Selective, and Bioavailable 5-HT2A Receptor Antagonists; J. Med. Chem., 2002, 45, 492-503.
4. Hutson, P. H.; Barton, C. L.; Jay, M.; Blurton, P.; Burkamp, F.; Clarkson, R.; Bristow, L. J.: Activation of mesolimbic dopamine function by phencyclidine is enhanced by 5-HT2C/2B receptor blockade: Neurochemical and behavioural studies; Neuropharm., 2000, 39, 2318-2328.
5. Enders, D.; Burkamp, F.; Runsink, J.: Diastereo- and enantioselective synthesis of 6-hetero substituted 3,5-dihydroxy esters: novel precursors of mevinolin analogs; Chem. Commun., 1996, 5, 609-610.
6. Enders, D.; Piva, O.; Burkamp, F.: Asymmetric synthesis of vicinal thioether alcohols by diastereoselective 1,2-addition of carbon nucleophiles to enantiomerically enriched -sulfenylated aldehydes; Tetrahedron, 1996, 52, 2893-2908.
7. Enders, D.; Lohray, B. B.; Burkamp, F.; Bhushan, V.; Hett, R.: Regio- and enantioselective synthesis of -silyl aldehydes and ketones via SAMP/RAMP hydrazones; Liebigs Ann., 1996, 2, 189-200.

History

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